Invention Grant
US08455550B2 Derivatives of aminocyclobutane or aminocyclobutene, their method of preparation and their use as medical products
有权
氨基环丁烷或氨基环丁烯的衍生物,其制备方法及其用作医药产品
- Patent Title: Derivatives of aminocyclobutane or aminocyclobutene, their method of preparation and their use as medical products
- Patent Title (中): 氨基环丁烷或氨基环丁烯的衍生物,其制备方法及其用作医药产品
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Application No.: US13258546Application Date: 2010-04-02
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Publication No.: US08455550B2Publication Date: 2013-06-04
- Inventor: Stéphane Cuisiat , Adrian Newman-Tancredi , Olivier Vitton , Bernard Vacher
- Applicant: Stéphane Cuisiat , Adrian Newman-Tancredi , Olivier Vitton , Bernard Vacher
- Applicant Address: FR Boulogne-Billancourt
- Assignee: Pierre Fabre Medicament
- Current Assignee: Pierre Fabre Medicament
- Current Assignee Address: FR Boulogne-Billancourt
- Agency: Birch, Stewart, Kolasch & Birch, LLP
- Priority: FR0952196 20090403
- International Application: PCT/EP2010/054452 WO 20100402
- International Announcement: WO2010/112597 WO 20101007
- Main IPC: A61K31/165
- IPC: A61K31/165 ; A61P25/00 ; C07C237/24

Abstract:
The present invention concerns compounds of general formula (1), where in:—-a- is a single or double bond, Ar is an aromatic group, substituted or unsubstituted, R1 and R2 each independently or together are: a hydrogen atom or C1-C6 alkyl group, branched or unbranched, saturated or unsaturated, substituted or unsubstituted; the groups R1 and R2 may also form a heterocycle, R3 and R3′ each independently or together are a hydrogen atom or C1-C6 alkyl group, X is an oxygen atom or a sulphur atom, and the addition salts of the compounds of general formula (1) with pharmaceutically acceptable mineral acids or organic acids.
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