Invention Grant
US08481584B2 1H-thieno[2,3-c]pyrazole derivatives useful as kinase inhibitors
失效
可用作激酶抑制剂的1H-噻吩并[2,3-c]吡唑衍生物
- Patent Title: 1H-thieno[2,3-c]pyrazole derivatives useful as kinase inhibitors
- Patent Title (中): 可用作激酶抑制剂的1H-噻吩并[2,3-c]吡唑衍生物
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Application No.: US13404697Application Date: 2012-02-24
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Publication No.: US08481584B2Publication Date: 2013-07-09
- Inventor: Daniele Fancelli , Paola Vianello , Mario Varasi , Simona Bindi , Sergio Vioglio , Dania Tesei
- Applicant: Daniele Fancelli , Paola Vianello , Mario Varasi , Simona Bindi , Sergio Vioglio , Dania Tesei
- Applicant Address: IT Nerviano (MI)
- Assignee: Nerviano Medical Sciences S.R.L.
- Current Assignee: Nerviano Medical Sciences S.R.L.
- Current Assignee Address: IT Nerviano (MI)
- Agency: Scully, Scott, Murphy & Presser, P.C.
- Main IPC: A61K31/4162
- IPC: A61K31/4162 ; C07D231/26
![1H-thieno[2,3-c]pyrazole derivatives useful as kinase inhibitors](/abs-image/US/2013/07/09/US08481584B2/abs.jpg.150x150.jpg)
Abstract:
Thieno[2,3-c]pyrazole derivatives of formula (I) and pharmaceutically acceptable salts thereof, as defined in the specification, process for their preparation and pharmaceutical compositions comprising them are disclosed; the compounds of the invention may be useful, in therapy, in the treatment of diseases associated with a disregulated protein kinase activity, like cancer.
Public/Granted literature
- US20120165311A1 1H-THIENO[2,3-C]PYRAZOLE DERIVATIVES USEFUL AS KINASE INHIBITORS Public/Granted day:2012-06-28
Information query
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