Invention Grant
- Patent Title: Phenylpropionamide compounds and the use thereof
- Patent Title (中): 苯丙酰胺化合物及其用途
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Application No.: US12447758Application Date: 2007-10-31
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Publication No.: US08481743B2Publication Date: 2013-07-09
- Inventor: Xiaoming Zhou
- Applicant: Xiaoming Zhou
- Applicant Address: US CT Stamford
- Assignee: Purdue Pharma L.P.
- Current Assignee: Purdue Pharma L.P.
- Current Assignee Address: US CT Stamford
- Agency: Purdue Pharma L.P.
- Agent Marian E. Fundytus; Alan L. Koller
- International Application: PCT/IB2007/003411 WO 20071031
- International Announcement: WO2008/053352 WO 20080508
- Main IPC: C07D211/56
- IPC: C07D211/56 ; A61K31/445
Abstract:
The invention relates to phenylpropionamide compounds of Formula (I): and pharmaceutically acceptable salts, prodrugs, and solvates thereof, wherein A, B, R1, R2, R3, R4 and R5 are defined as set forth in the specification. The invention is also directed to the use of compounds of Formula (I) to treat, prevent or ameliorate a disorder responsive to the activation of opioid receptors, particularly μ-opioid receptors. Compounds of the present invention are especially useful for treating pain.
Public/Granted literature
- US20100234426A1 Phenylpropionamide Compounds and the Use Thereof Public/Granted day:2010-09-16
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