Invention Grant
- Patent Title: Self-microemulsifying mitotane composition
- Patent Title (中): 自我微乳化米托坦组合物
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Application No.: US13322222Application Date: 2010-05-24
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Publication No.: US08486445B2Publication Date: 2013-07-16
- Inventor: Florian Battung , Emad Hassan , Lionel Sansoe
- Applicant: Florian Battung , Emad Hassan , Lionel Sansoe
- Agency: Saliwanchik, Lloyd & Eisenschenk
- Priority: EP09160999 20090525
- International Application: PCT/IB2010/052292 WO 20100524
- International Announcement: WO2010/136952 WO 20101202
- Main IPC: A61K9/107
- IPC: A61K9/107 ; A61K9/113 ; A61K9/48 ; A61K31/02

Abstract:
The invention relates to a self-microemulsifying drug delivery system (“SMEDDS”) of mitotane, with enhanced bioavailability. More particularly the invention provides a mitotane oily formulation comprising propylene glycol monocaprylate (10 to 30% w/w), propylene glycol dicaprate (20 to 60% w/w) and polyoxyethylenesorbitanne monooleate (10 to 30% w/w).
Public/Granted literature
- US20130017258A1 SELF-MICROEMULSIFYING MITOTANE COMPOSITION Public/Granted day:2013-01-17
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