Invention Grant
- Patent Title: Macrocyclic integrase inhibitors
- Patent Title (中): 大环整合酶抑制剂
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Application No.: US13395891Application Date: 2010-10-13
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Publication No.: US08497270B2Publication Date: 2013-07-30
- Inventor: Johannes Wilhelmus J Thuring , Jean-Francois Bonfanti , Jerome Michel Claude Fortin
- Applicant: Johannes Wilhelmus J Thuring , Jean-Francois Bonfanti , Jerome Michel Claude Fortin
- Applicant Address: US IN Indianapolis
- Assignee: Elanco Animal Health Ireland Limited
- Current Assignee: Elanco Animal Health Ireland Limited
- Current Assignee Address: US IN Indianapolis
- Agent James J. Sales
- Priority: EP09172853 20091013
- International Application: PCT/EP2010/065300 WO 20101013
- International Announcement: WO2011/045330 WO 20110421
- Main IPC: C07D471/18
- IPC: C07D471/18 ; C07D498/18 ; C07D513/18 ; C07D515/18 ; C07D498/22 ; A61K31/547 ; A61P31/18
Abstract:
Compound having formula (I), wherein —W is NH—, —N(CH3)— or piperazine, —X is a bond, —C(═O)— or S(═O)2—, —Y is C3-7alkylene, and —Z is NH—C(═O)— or —O—, and pharmaceutically acceptable salts thereof, their pharmaceutical formulations and use as HIV inhibitors.
Public/Granted literature
- US20120172367A1 MACROCYCLIC INTEGRASE INHIBITORS Public/Granted day:2012-07-05
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