Invention Grant
US08524728B2 Substituted indolyl alkyl amino derivatives as novel inhibitors of histone deacetylase
有权
取代的吲哚基烷基氨基衍生物作为组蛋白脱乙酰酶的新型抑制剂
- Patent Title: Substituted indolyl alkyl amino derivatives as novel inhibitors of histone deacetylase
- Patent Title (中): 取代的吲哚基烷基氨基衍生物作为组蛋白脱乙酰酶的新型抑制剂
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Application No.: US13027793Application Date: 2011-02-15
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Publication No.: US08524728B2Publication Date: 2013-09-03
- Inventor: Marc Gustaaf Celine Verdonck , Patrick René Angibaud , Bruno Roux , Isabelle Noëlle Constance Pilatte , Peter Ten Holte , Janine Arts , Kristof Van Emelen
- Applicant: Marc Gustaaf Celine Verdonck , Patrick René Angibaud , Bruno Roux , Isabelle Noëlle Constance Pilatte , Peter Ten Holte , Janine Arts , Kristof Van Emelen
- Applicant Address: BE Beerse
- Assignee: Janssen Pharmaceutica N.V.
- Current Assignee: Janssen Pharmaceutica N.V.
- Current Assignee Address: BE Beerse
- Priority: EP04077172 20040728
- Main IPC: A61K31/506
- IPC: A61K31/506 ; C07D401/14
Abstract:
This invention comprises the novel compounds of formula (I) wherein R1, R2, R3, X and Y have defined meanings, having histone deacetylase inhibiting enzymatic activity; their preparation, compositions containing them and their use as a medicine.
Public/Granted literature
- US20110136841A1 SUBSTITUTED INDOLYL ALKYL AMINO DERIVATIVES AS NOVEL INHIBITORS OF HISTONE DEACETYLASE Public/Granted day:2011-06-09
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