Invention Grant
US08575199B2 Formula (IA″) compounds comprising (piperidin-4-yl)pyridine or (1,2,3,6-tetrahydropyridin-4-4yl) as TRPV1 antagonists
有权
包含（哌啶-4-基）吡啶或（1,2,3,6-四氢吡啶-4- 4-基）作为TRPV1拮抗剂的式（IA“）化合物
- Patent Title: Formula (IA″) compounds comprising (piperidin-4-yl)pyridine or (1,2,3,6-tetrahydropyridin-4-4yl) as TRPV1 antagonists
- Patent Title (中): 包含（哌啶-4-基）吡啶或（1,2,3,6-四氢吡啶-4- 4-基）作为TRPV1拮抗剂的式（IA“）化合物
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Application No.: US13396450Application Date: 2012-02-14
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Publication No.: US08575199B2Publication Date: 2013-11-05
- Inventor: Laykea Tafesse
- Applicant: Laykea Tafesse
- Applicant Address: US CT Stamford
- Assignee: Purdue Pharma L.P.
- Current Assignee: Purdue Pharma L.P.
- Current Assignee Address: US CT Stamford
- Agency: Dechert LLP
- Main IPC: A61K31/44
- IPC: A61K31/44
Abstract:
The invention relates to compounds of formula IA″ and pharmaceutically acceptable derivatives thereof, compositions comprising an effective amount of a compound of formula IA″ or a pharmaceutically acceptable derivative thereof, and methods for treating or preventing a condition such as pain, UI, an ulcer, IBD and IBS, comprising administering to an animal in need thereof an effective amount of a compound of formula IA″ or a pharmaceutically acceptable derivative thereof.
Public/Granted literature
- US20120177570A1 TRPV1 ANTAGONISTS INCLUDING AMIDE SUBSTITUENT AND USES THEREOF Public/Granted day:2012-07-12
Information query
