Invention Grant
- Patent Title: Heterocyclic amides as modulators of TRPA1
- Patent Title (中): 杂环酰胺作为TRPA1的调节剂
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Application No.: US13375833Application Date: 2010-06-04
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Publication No.: US08614201B2Publication Date: 2013-12-24
- Inventor: Didier Jean-Calude Berthelot , Henricus Jacobus Maria Gijsen , Mirko Zaja , Jason Rech , Alec Lebsack , Bryan Branstetter , Wei Xiao , J. Guy Breitenbucher
- Applicant: Didier Jean-Calude Berthelot , Henricus Jacobus Maria Gijsen , Mirko Zaja , Jason Rech , Alec Lebsack , Bryan Branstetter , Wei Xiao , J. Guy Breitenbucher
- Applicant Address: BE Beerse
- Assignee: Janssen Pharmaceutica NV
- Current Assignee: Janssen Pharmaceutica NV
- Current Assignee Address: BE Beerse
- International Application: PCT/US2010/037381 WO 20100604
- International Announcement: WO2010/141805 WO 20101209
- Main IPC: A01N57/00
- IPC: A01N57/00 ; A61K31/66 ; A01N43/36 ; A61K31/40 ; A01N43/66 ; A61K31/53 ; A01N43/40 ; A61K31/435 ; A01N43/54 ; C07D239/42 ; C07D401/04 ; C07D239/00 ; C07D239/02 ; C07D213/00 ; C07C303/00 ; C07C307/00 ; C07C309/00 ; C07C311/00

Abstract:
Certain heterocyclic amide compounds are described. The compounds may be used in pharmaceutical compositions and methods for treating disease states, disorders, and conditions mediated by TRPA1 activity, such as pain, arthritis, itch, cough, asthma, or inflammatory bowel disease.
Public/Granted literature
- US20120083474A1 HETEROCYCLIC AMIDES AS MODULATORS OF TRPA1 Public/Granted day:2012-04-05
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