Invention Grant
- Patent Title: Quinazolinone derivatives as PARP inhibitors
- Patent Title (中): 喹唑啉酮衍生物作为PARP抑制剂
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Application No.: US11569892Application Date: 2005-06-28
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Publication No.: US08623872B2Publication Date: 2014-01-07
- Inventor: Jérôme Emile Georges Guillemont , Ludo Edmond Josephine Kennis , Josephus Carolus Mertens , Jacobus Alphonsus Josephus Van Dun , Maria Victorina Francisca Somers , Walter Boudewijn Leopold Wouters
- Applicant: Jérôme Emile Georges Guillemont , Ludo Edmond Josephine Kennis , Josephus Carolus Mertens , Jacobus Alphonsus Josephus Van Dun , Maria Victorina Francisca Somers , Walter Boudewijn Leopold Wouters
- Applicant Address: BE
- Assignee: Janssen Pharmaceutica, NV
- Current Assignee: Janssen Pharmaceutica, NV
- Current Assignee Address: BE
- Priority: EP04076887 20040630
- International Application: PCT/EP2005/053029 WO 20050628
- International Announcement: WO2006/003146 WO 20060112
- Main IPC: A61K31/497
- IPC: A61K31/497 ; C07D239/72

Abstract:
The present invention provides compounds of formula (I), their use as PARP inhibitors as well as pharmaceutical compositions comprising said compounds of formula (I) wherein R1, R2, R3, L, X, Y and Z have defined meanings.
Public/Granted literature
- US20080070915A1 Quinazoline Derivatives as Parp Inhibitors Public/Granted day:2008-03-20
Information query
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