Invention Grant
US08648063B2 Potentiation of cancer chemotherapy by 7-(2, 5-dihydro-4-imidazo [1, 2-a] pyridine-3-yl-2,5-dioxo-1H-pyrrol-3-yl)-9-fluoro-1,2,3,4 tetrahydro -2-(1-piperidinyl-carbonyl)-pyrrolo [3,2,1-jk] [1,4] benzodiazepine 失效
7-(2,5-二氢-4-咪唑并[1,2-a]吡啶-3-基-2,5-二氧代-1H-吡咯-3-基)-9-氟-1 ,2,3,4四氢-2-(1-哌啶基 - 羰基) - 吡咯并[3,2,1-jk] [1,4]苯并二氮杂

  • Patent Title: Potentiation of cancer chemotherapy by 7-(2, 5-dihydro-4-imidazo [1, 2-a] pyridine-3-yl-2,5-dioxo-1H-pyrrol-3-yl)-9-fluoro-1,2,3,4 tetrahydro -2-(1-piperidinyl-carbonyl)-pyrrolo [3,2,1-jk] [1,4] benzodiazepine
  • Patent Title (中): 7-(2,5-二氢-4-咪唑并[1,2-a]吡啶-3-基-2,5-二氧代-1H-吡咯-3-基)-9-氟-1 ,2,3,4四氢-2-(1-哌啶基 - 羰基) - 吡咯并[3,2,1-jk] [1,4]苯并二氮杂
  • Application No.: US13654884
    Application Date: 2012-10-18
  • Publication No.: US08648063B2
    Publication Date: 2014-02-11
  • Inventor: Marcio ChedidThomas Albert Engler
  • Applicant: Eli Lilly and Company
  • Applicant Address: US IN Indianapolis
  • Assignee: Eli Lilly and Company
  • Current Assignee: Eli Lilly and Company
  • Current Assignee Address: US IN Indianapolis
  • Agent John C Demeter; Robert D Titus
  • Main IPC: A01N43/00
  • IPC: A01N43/00 A61K31/33 A01N43/62 A61K31/55
Potentiation of cancer chemotherapy by 7-(2, 5-dihydro-4-imidazo [1, 2-a] pyridine-3-yl-2,5-dioxo-1H-pyrrol-3-yl)-9-fluoro-1,2,3,4 tetrahydro -2-(1-piperidinyl-carbonyl)-pyrrolo [3,2,1-jk] [1,4] benzodiazepine
Abstract:
An improved method for treating gastric cancer, ovarian cancer, non-small cell lung cancer, or colorectal cancer in a patient is described, as well as pharmaceutical compositions useful for the method and a process for preparing said compositions.
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