Invention Grant
US08648063B2 Potentiation of cancer chemotherapy by 7-(2, 5-dihydro-4-imidazo [1, 2-a] pyridine-3-yl-2,5-dioxo-1H-pyrrol-3-yl)-9-fluoro-1,2,3,4 tetrahydro -2-(1-piperidinyl-carbonyl)-pyrrolo [3,2,1-jk] [1,4] benzodiazepine
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7-(2,5-二氢-4-咪唑并[1,2-a]吡啶-3-基-2,5-二氧代-1H-吡咯-3-基)-9-氟-1 ,2,3,4四氢-2-(1-哌啶基 - 羰基) - 吡咯并[3,2,1-jk] [1,4]苯并二氮杂
- Patent Title: Potentiation of cancer chemotherapy by 7-(2, 5-dihydro-4-imidazo [1, 2-a] pyridine-3-yl-2,5-dioxo-1H-pyrrol-3-yl)-9-fluoro-1,2,3,4 tetrahydro -2-(1-piperidinyl-carbonyl)-pyrrolo [3,2,1-jk] [1,4] benzodiazepine
- Patent Title (中): 7-(2,5-二氢-4-咪唑并[1,2-a]吡啶-3-基-2,5-二氧代-1H-吡咯-3-基)-9-氟-1 ,2,3,4四氢-2-(1-哌啶基 - 羰基) - 吡咯并[3,2,1-jk] [1,4]苯并二氮杂
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Application No.: US13654884Application Date: 2012-10-18
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Publication No.: US08648063B2Publication Date: 2014-02-11
- Inventor: Marcio Chedid , Thomas Albert Engler
- Applicant: Eli Lilly and Company
- Applicant Address: US IN Indianapolis
- Assignee: Eli Lilly and Company
- Current Assignee: Eli Lilly and Company
- Current Assignee Address: US IN Indianapolis
- Agent John C Demeter; Robert D Titus
- Main IPC: A01N43/00
- IPC: A01N43/00 ; A61K31/33 ; A01N43/62 ; A61K31/55
![Potentiation of cancer chemotherapy by 7-(2, 5-dihydro-4-imidazo [1, 2-a] pyridine-3-yl-2,5-dioxo-1H-pyrrol-3-yl)-9-fluoro-1,2,3,4 tetrahydro -2-(1-piperidinyl-carbonyl)-pyrrolo [3,2,1-jk] [1,4] benzodiazepine](/abs-image/US/2014/02/11/US08648063B2/abs.jpg.150x150.jpg)
Abstract:
An improved method for treating gastric cancer, ovarian cancer, non-small cell lung cancer, or colorectal cancer in a patient is described, as well as pharmaceutical compositions useful for the method and a process for preparing said compositions.
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