Invention Grant
- Patent Title: Anti-misuse microparticulate oral pharmaceutical form
- Patent Title (中): 反滥用微粒口服药物形式
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Application No.: US11439432Application Date: 2006-05-24
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Publication No.: US08652529B2Publication Date: 2014-02-18
- Inventor: Florence Guimberteau , Frédéric Dargelas
- Applicant: Florence Guimberteau , Frédéric Dargelas
- Applicant Address: FR Venissieux
- Assignee: Flamel Technologies
- Current Assignee: Flamel Technologies
- Current Assignee Address: FR Venissieux
- Agency: Patton Boggs LLP
- Priority: FR0553437 20051110
- Main IPC: A61K9/16
- IPC: A61K9/16

Abstract:
The present invention relates to solid microparticulate oral pharmaceutical forms whose composition and structure make it possible to avoid misuse of the pharmaceutical active principle they contain. The invention relates to a solid oral pharmaceutical form which is characterized in that it contains anti-misuse means, in that at least part of the active principle it comprises is contained in coated microparticles for modified release of the active principle, and in that the coated microparticles have a coating layer which assures modified release of the active principle and simultaneously imparts crushing resistance to the coated microparticles so as to avoid misuse.
Public/Granted literature
- US20070224129A1 Anti-misuse microparticulate oral pharmaceutical form Public/Granted day:2007-09-27
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