Invention Grant
- Patent Title: Process for the preparation of asenapine
- Patent Title (中): 制备阿替那平的方法
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Application No.: US13812212Application Date: 2011-07-29
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Publication No.: US08653280B2Publication Date: 2014-02-18
- Inventor: Pere Dalmases Barjoan , Juan Huguet Clotet , Jordi Peirats Masia
- Applicant: Pere Dalmases Barjoan , Juan Huguet Clotet , Jordi Peirats Masia
- Applicant Address: ES Sant Joan Despi
- Assignee: Laboratories Lesvi, S.L.
- Current Assignee: Laboratories Lesvi, S.L.
- Current Assignee Address: ES Sant Joan Despi
- Agency: Barnes & Thornburg LLP
- Priority: EP10171222 20100729
- International Application: PCT/EP2011/063071 WO 20110729
- International Announcement: WO2012/013766 WO 20120202
- Main IPC: C07D491/044
- IPC: C07D491/044 ; C07D313/14
Abstract:
The present invention is directed to novel compounds of formula (I) as well as to the process for their preparation. Novel compounds of formula (I) can be converted into asenapine through an efficient process. The invention also relates to novel intermediates used in this process and their use in the preparation of compounds of formula (I).
Public/Granted literature
- US20130225835A1 NOVEL PROCESS FOR THE PREPARATION OF ASENAPINE Public/Granted day:2013-08-29
Information query
