Invention Grant
- Patent Title: Solid forms of an azocyclic amide
- Patent Title (中): 固体形式的杂环酰胺
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Application No.: US13265138Application Date: 2010-04-19
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Publication No.: US08669277B2Publication Date: 2014-03-11
- Inventor: Matthew Richard Oberholzer , Robert James Pasteris , Rafael Shapiro
- Applicant: Matthew Richard Oberholzer , Robert James Pasteris , Rafael Shapiro
- Applicant Address: US DE Wilmington
- Assignee: E I du Pont de Nemours and Company
- Current Assignee: E I du Pont de Nemours and Company
- Current Assignee Address: US DE Wilmington
- Agent Renee M. Lett
- International Application: PCT/US2010/031546 WO 20100419
- International Announcement: WO2010/123791 WO 20101028
- Main IPC: A61K31/454
- IPC: A61K31/454 ; C07D417/14

Abstract:
Disclosed are solid forms of 1-[4-[4-[5-(2,6-difluorophenyl)-4,5-dihydro-3-isoxazolyl]-2-thiazolyl]-1-piperidinyl]-2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethanone (Compound 1). Methods for the preparation of solid forms of Compound 1 and for the conversion of one solid form of Compound 1 into another are disclosed.Disclosed are fungicidal compositions comprising a fungicidally effective amount of a solid form of Compound 1 and at least one additional component selected from the group consisting of surfactants, solid diluents and liquid carriers. Compositions comprising a mixture of a solid form of Compound 1 and at least one other fungicide or insecticide are also disclosed.Also disclosed are methods for controlling plant diseases caused by fungal plant pathogens comprising applying to a plant or portion thereof, or to a plant seed, a fungicidally effective amount of a solid form of Compound 1.
Public/Granted literature
- US20120034315A1 SOLID FORMS OF AN AZOCYCLIC AMIDE Public/Granted day:2012-02-09
Information query
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