Invention Grant
- Patent Title: Process for preparing aminobenzofuran derivatives
- Patent Title (中): 制备氨基苯并呋喃衍生物的方法
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Application No.: US13628867Application Date: 2012-09-27
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Publication No.: US08686180B2Publication Date: 2014-04-01
- Inventor: Xavier Bon , Corinne Leroy
- Applicant: SANOFI
- Applicant Address: FR Paris
- Assignee: SANOFI
- Current Assignee: SANOFI
- Current Assignee Address: FR Paris
- Agency: Scully, Scott, Murphy & Presser, P.C.
- Priority: FR1052481 20100401
- Main IPC: C07C229/00
- IPC: C07C229/00

Abstract:
This disclosure relates to a process for preparing 5-aminobenzofuran derivatives of general formula (I): in which R1 and R2 are as defined in the description, by treating a 5-N-alkylamidobenzofuran derivative of general formula (II): in which R1, R2, and R3 are as defined in the description, with a strong acid, so as to form an acid addition salt of the compound of formula (I), which salt is itself treated, if necessary, with a basic agent so as to form this compound of formula (I) in free base form.
Public/Granted literature
- US20130023677A1 PROCESS FOR PREPARING AMINOBENZOFURAN DERIVATIVES Public/Granted day:2013-01-24
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