Invention Grant
US08691860B2 Crystals and process of making 5-({(2-amino-3-(4-carbamoyl-2,6-dimethyl-phenyl)-propionyl]-[1-(-4-phenyl-1h-imidazol-2-yl)-ethyl]-amino}-methyl)-2-methoxy-benzoic acid
有权
制备5 - （{（2-氨基-3-（4-氨基甲酰基-2,6-二甲基 - 苯基） - 丙酰基] - [1-（4-苯基-1H-咪唑-2-基） 乙基] - 氨基} - 甲基）-2-甲氧基 - 苯甲酸
![Crystals and process of making 5-({(2-amino-3-(4-carbamoyl-2,6-dimethyl-phenyl)-propionyl]-[1-(-4-phenyl-1h-imidazol-2-yl)-ethyl]-amino}-methyl)-2-methoxy-benzoic acid](/docs/US/2014-04-08/US08691860B2/abs.jpg.600x600.jpg)
- Patent Title: Crystals and process of making 5-({(2-amino-3-(4-carbamoyl-2,6-dimethyl-phenyl)-propionyl]-[1-(-4-phenyl-1h-imidazol-2-yl)-ethyl]-amino}-methyl)-2-methoxy-benzoic acid
- Patent Title (中): 制备5 - （{（2-氨基-3-（4-氨基甲酰基-2,6-二甲基 - 苯基） - 丙酰基] - [1-（4-苯基-1H-咪唑-2-基） 乙基] - 氨基} - 甲基）-2-甲氧基 - 苯甲酸
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Application No.: US13987009Application Date: 2013-06-24
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Publication No.: US08691860B2Publication Date: 2014-04-08
- Inventor: Luigi Anzalone , Frank J. Villani , Christopher A. Teleha , Penina Feibush , Barry Fegely
- Applicant: Furiex Pharmaceuticals, Inc.
- Applicant Address: US NC Morrisville
- Assignee: Furiex Pharmaceuticals, Inc.
- Current Assignee: Furiex Pharmaceuticals, Inc.
- Current Assignee Address: US NC Morrisville
- Agency: Sheridan Ross P.C.
- Main IPC: A61K31/4164
- IPC: A61K31/4164 ; C07D233/64
![Crystals and process of making 5-({(2-amino-3-(4-carbamoyl-2,6-dimethyl-phenyl)-propionyl]-[1-(-4-phenyl-1h-imidazol-2-yl)-ethyl]-amino}-methyl)-2-methoxy-benzoic acid](/abs-image/US/2014/04/08/US08691860B2/abs.jpg.150x150.jpg)
Abstract:
The present invention relates to a novel crystals of 5-({[2-amino-3-(4-carbamoyl-2,6-dimethyl-phenyl)-propionyl]-[1-(4-phenyl-1h-imidazol-2-yl)-ethyl]-amino}-methyl)-2-methoxy-benzoic acid and methods of making the zwitterion of 5-({[2-amino-3-(4-carbamoyl-2,6-dimethyl-phenyl)-propionyl]-[1-(4-phenyl-1h-imidazol-2-yl)-ethyl]-amino}-methyl)-2-methoxy-benzoic acid.
Public/Granted literature
- US20140011851A1 Novel crystals and process of making 5-(-METHYL)-2-METHOXY-BENZOIC ACID Public/Granted day:2014-01-09
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