Invention Grant
US08697700B2 Piperazinone-substituted tetrahydro-carboline MCH-1 antagonists, methods of making, and uses thereof
失效
哌嗪酮取代的四氢 - 咔啉MCH-1拮抗剂，其制备方法和用途
- Patent Title: Piperazinone-substituted tetrahydro-carboline MCH-1 antagonists, methods of making, and uses thereof
- Patent Title (中): 哌嗪酮取代的四氢 - 咔啉MCH-1拮抗剂，其制备方法和用途
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Application No.: US13330989Application Date: 2011-12-20
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Publication No.: US08697700B2Publication Date: 2014-04-15
- Inventor: Matthew D. Surman , Peter R. Guzzo
- Applicant: Matthew D. Surman , Peter R. Guzzo
- Applicant Address: US NY Albany
- Assignee: Albany Molecular Research, Inc.
- Current Assignee: Albany Molecular Research, Inc.
- Current Assignee Address: US NY Albany
- Agency: LeClairRyan
- Main IPC: A61K31/496
- IPC: A61K31/496 ; A61K31/501 ; A61K31/506 ; C07D471/04
Abstract:
The present invention relates to piperazinone-substituted tetrahydrocarboline derivatives of formula (I): having the substituents as described herein which are melanin-concentrating hormone (MCH-1) receptor antagonists. The present invention also relates to pharmaceutical compositions including these compounds, and methods of preparation and use thereof.
Public/Granted literature
- US20120157469A1 PIPERAZINONE-SUBSTITUTED TETRAHYDRO-CARBOLINE MCH-1 ANTAGONISTS, METHODS OF MAKING, AND USES THEREOF Public/Granted day:2012-06-21
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