Invention Grant
- Patent Title: Glycine transporter inhibiting substances
- Patent Title (中): 甘氨酸转运蛋白抑制物质
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Application No.: US13823574Application Date: 2011-09-16
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Publication No.: US08729271B2Publication Date: 2014-05-20
- Inventor: Minoru Moriya , Akito Yasuhara , Kazunari Sakagami , Hiroshi Ohta , Kumi Abe , Shuji Yamamoto , Yuko Araki , Hiroki Urabe , Xiang-Min Sun
- Applicant: Minoru Moriya , Akito Yasuhara , Kazunari Sakagami , Hiroshi Ohta , Kumi Abe , Shuji Yamamoto , Yuko Araki , Hiroki Urabe , Xiang-Min Sun
- Applicant Address: JP Tokyo
- Assignee: Taisho Pharmaceutical Co., Ltd
- Current Assignee: Taisho Pharmaceutical Co., Ltd
- Current Assignee Address: JP Tokyo
- Agency: Sughrue Mion, PLLC
- Priority: JP2010-209184 20100917
- International Application: PCT/JP2011/071241 WO 20110916
- International Announcement: WO2012/036278 WO 20120322
- Main IPC: A01N43/40
- IPC: A01N43/40 ; A61K31/44 ; A01N43/64 ; A61K31/41 ; C07D213/00 ; C07D401/00 ; C07D419/00

Abstract:
The present invention aims to provide novel compounds of formula [I] or pharmaceutically acceptable salts thereof that are based on a glycine uptake inhibiting action and which are useful in the prevention or treatment of such diseases as schizophrenia, Alzheimer's disease, cognitive dysfunction, dementia, anxiety disorders (generalized anxiety disorder, panic disorder, obsessive-compulsive disorder, social anxiety disorder, posttraumatic stress disorder, specific phobia, acute stress disorder, etc.), depression, drug addiction, spasm, tremor, pain, and sleep disorder:
Public/Granted literature
- US20130184460A1 GLYCINE TRANSPORTER INHIBITING SUBSTANCES Public/Granted day:2013-07-18
Information query
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