Invention Grant
US08735408B2 Solid forms of 3-(4-(aminomethyl)-1-(5-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperidine-4-carboxamido)phenyl dimethylcarbamate
有权
固体形式的3-(4-(氨基甲基)-1-(5-甲基-7H-吡咯并[2,3-d]嘧啶-4-基)哌啶-4-甲酰氨基)苯基二甲基氨基甲酸酯
- Patent Title: Solid forms of 3-(4-(aminomethyl)-1-(5-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperidine-4-carboxamido)phenyl dimethylcarbamate
- Patent Title (中): 固体形式的3-(4-(氨基甲基)-1-(5-甲基-7H-吡咯并[2,3-d]嘧啶-4-基)哌啶-4-甲酰氨基)苯基二甲基氨基甲酸酯
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Application No.: US13288321Application Date: 2011-11-03
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Publication No.: US08735408B2Publication Date: 2014-05-27
- Inventor: Susan Margaret De Paul , Qun Li , Haiming Zhang
- Applicant: Susan Margaret De Paul , Qun Li , Haiming Zhang
- Applicant Address: US TX The Woodlands
- Assignee: Lexicon Pharmaceuticals, Inc.
- Current Assignee: Lexicon Pharmaceuticals, Inc.
- Current Assignee Address: US TX The Woodlands
- Agent Max Bachrach
- Main IPC: C07D487/04
- IPC: C07D487/04 ; A61K31/519 ; A61P27/06
![Solid forms of 3-(4-(aminomethyl)-1-(5-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperidine-4-carboxamido)phenyl dimethylcarbamate](/abs-image/US/2014/05/27/US08735408B2/abs.jpg.150x150.jpg)
Abstract:
Solid forms of 3-(4-(aminomethyl)-1-(5-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)piperidine-4-carboxamido)phenyl dimethylcarbamate and salts thereof are disclosed. Methods of its use to treat diseases and disorders of the eye are also disclosed.
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