Invention Grant
- Patent Title: Compounds
- Patent Title (中): 化合物
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Application No.: US13897853Application Date: 2013-05-20
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Publication No.: US08742099B2Publication Date: 2014-06-03
- Inventor: Alan David Borthwick , Deirdre Mary Bernadette Hickey , John Liddle , Andrew McMurtrie Mason
- Applicant: Glaxo Group Limited
- Applicant Address: GB Brentford, Middlesex
- Assignee: Glaxo Group Limited
- Current Assignee: Glaxo Group Limited
- Current Assignee Address: GB Brentford, Middlesex
- Agent Kathryn L. Coulter
- Priority: GB0414093.5 20040623
- Main IPC: C07D413/14
- IPC: C07D413/14

Abstract:
Compounds of formula (I) wherein R1 is 2-indanyl, R2 is 1-methylpropyl, R3 is a group selected from 2,6-dimethyl-3-pyridyl or 4,6-dimethyl-3-pyridyl, R4 represents methyl and R5 represents hydrogen or methyl or, R4 and R5 together with the nitrogen atom to which they are attached represent morpholino and pharmaceutically acceptable derivatives thereof are described, as are processes for their preparation, pharmaceutical compositions containing them and their use in medicine, particularly their use as oxytocin antagonists.
Public/Granted literature
- US20130253188A1 NOVEL COMPOUNDS Public/Granted day:2013-09-26
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