Invention Grant
- Patent Title: Furanone derivative
- Patent Title (中): 呋喃酮衍生物
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Application No.: US14008488Application Date: 2012-03-30
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Publication No.: US08742113B2Publication Date: 2014-06-03
- Inventor: Takayuki Irie , Ayako Sawa , Masaaki Sawa , Tokiko Asami , Yoko Funakoshi , Chika Tanaka
- Applicant: Takayuki Irie , Ayako Sawa , Masaaki Sawa , Tokiko Asami , Yoko Funakoshi , Chika Tanaka
- Applicant Address: JP Tokyo JP Kobe-shi
- Assignee: SBI Biotech Co., Ltd.,Carna Biosciences, Inc.
- Current Assignee: SBI Biotech Co., Ltd.,Carna Biosciences, Inc.
- Current Assignee Address: JP Tokyo JP Kobe-shi
- Agency: Westerman, Hattori, Daniels & Adrian, LLP
- Priority: JP2011-080185 20110331
- International Application: PCT/JP2012/058636 WO 20120330
- International Announcement: WO2012/113802 WO 20121004
- Main IPC: C07D471/02
- IPC: C07D471/02 ; C07D491/02 ; C07D498/02 ; C07D513/02 ; C07D515/02

Abstract:
To provide a novel furanone derivative, and a medicine including the same. The furanone derivative is represented by the formula (I): wherein A represents —COOR1 or a hydrogen atom; R1 represents a hydrogen atom, an optionally substituted hydrocarbon group, or an optionally substituted heterocycle; R2 and R3 are the same or different and each independently represent a hydrogen atom, an optionally substituted hydrocarbon group, an optionally substituted phenyl group, an optionally substituted heterocycle, an optionally substituted heterocyclic fused ring, or an optionally substituted amino group; or alternatively, R2 and R3, taken together with the nitrogen atom to which they are attached, may form an optionally substituted heterocycle or an optionally substituted heterocyclic fused ring; and R4 represents a hydrogen atom or a halogen atom; with the proviso that when A represents —COOR1, R2 and R3 are not optionally substituted amino groups at the same time, and when A represents a hydrogen atom, R3 represents a hydrogen atom.
Public/Granted literature
- US20140018533A1 NOVEL FURANONE DERIVATIVE Public/Granted day:2014-01-16
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