Invention Grant
- Patent Title: Quinuclidine esters of 1-azaheterocyclylacetic acid as antimuscarinic agents, process for their preparation and medicinal compositions thereof
- Patent Title (中): 1-氮杂环丁基乙酸的奎宁环酯作为抗毒蕈碱剂,其制备方法及其药用组合物
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Application No.: US13729388Application Date: 2012-12-28
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Publication No.: US08748613B2Publication Date: 2014-06-10
- Inventor: Gabriele Amari , Cristina Pesenti , Stefano Bossolo
- Applicant: Chiesi Farmaceutici S.p.A.
- Applicant Address: IT Parma
- Assignee: Chiesi Farmaceutici S.p.A.
- Current Assignee: Chiesi Farmaceutici S.p.A.
- Current Assignee Address: IT Parma
- Agency: Oblon, Spivak, McClelland, Maier & Neustadt, L.L.P.
- Priority: EP11196173 20111230
- Main IPC: A01N43/90
- IPC: A01N43/90 ; A01N43/40 ; A61K31/44 ; A61K31/445 ; C07D453/02 ; C07D211/00 ; C07D295/00 ; C07D401/00 ; C07D405/00

Abstract:
Compounds of formula (I): wherein A, R1, R2, X, m, and n are as defined in the specification, are selective M3 receptor antagonists and may be used in the treatment of, inter alia, a respiratory disease such as asthma and COPD.
Public/Granted literature
Information query
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