Invention Grant
- Patent Title: Solifenacin salts
- Patent Title (中): 索非那新盐
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Application No.: US13805828Application Date: 2011-07-05
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Publication No.: US08765785B2Publication Date: 2014-07-01
- Inventor: Gerardo Gutiérrez Fuentes , Antonio Lorente Bonde-Larsen , Jaime del Campo López-Bachiller , Celso Sandoval Rodríguez , Yolanda Fernández Sainz
- Applicant: Gerardo Gutiérrez Fuentes , Antonio Lorente Bonde-Larsen , Jaime del Campo López-Bachiller , Celso Sandoval Rodríguez , Yolanda Fernández Sainz
- Applicant Address: ES Boecillo
- Assignee: Crystal Pharma, S.A.U.
- Current Assignee: Crystal Pharma, S.A.U.
- Current Assignee Address: ES Boecillo
- Agency: Knobbe Martens Olson & Bear LLP
- Priority: EP10168415 20100705
- International Application: PCT/EP2011/061314 WO 20110705
- International Announcement: WO2012/004264 WO 20120112
- Main IPC: C07D453/02
- IPC: C07D453/02 ; A61K31/439

Abstract:
The invention concerns fumarate salts of solifenacin, as well as pharmaceutical compositions comprising fumarate salts of solifenacin. The invention furthermore concerns a process for preparing solifenacin and salts thereof. The fumarate salt provides improved properties over the known solifenacin salts, especially in terms of its stability. The novel process for its preparation is furthermore improved over known processes for preparing solifenacin in that it provides a higher yield and recovers a greater amount of starting material.
Public/Granted literature
- US20130203804A1 SOLIFENACIN SALTS Public/Granted day:2013-08-08
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