Invention Grant
- Patent Title: Trisubstituted 1,2,4 triazoles
- Patent Title (中): 三取代的1,2,4-三唑
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Application No.: US12866054Application Date: 2009-03-18
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Publication No.: US08778974B2Publication Date: 2014-07-15
- Inventor: Gregor James MacDonald , Johannes Wilhelmus John F. Thuring , Pauline Carol Stanislawski , Wei Zhuang , Yves Emiel Maria Van Roosbroeck , Frans Alfons Maria Van Den Keybus
- Applicant: Gregor James MacDonald , Johannes Wilhelmus John F. Thuring , Pauline Carol Stanislawski , Wei Zhuang , Yves Emiel Maria Van Roosbroeck , Frans Alfons Maria Van Den Keybus
- Applicant Address: BE Beerse
- Assignee: Janssen Pharmaceutica NV
- Current Assignee: Janssen Pharmaceutica NV
- Current Assignee Address: BE Beerse
- Agent Peter Herridge
- Priority: EP08152987 20080319
- International Application: PCT/EP2009/053186 WO 20090318
- International Announcement: WO2009/115547 WO 20090924
- Main IPC: A61K31/4439
- IPC: A61K31/4439 ; C07D401/04

Abstract:
The present invention relates to 1-aryl-3-aniline-5-alkyl-1,2,4-triazole derivatives and analogues or pharmaceutically acceptable salts thereof, processes for preparing them, pharmaceutical compositions containing them and their use in therapy, according to Formula (I).The invention particularly relates to potent positive allosteric modulators of nicotinic acetylcholine receptors, such positive allosteric modulator having the capability to increase the efficacy of nicotinic receptor agonists.
Public/Granted literature
- US20100324053A1 TRISUBSTITUTED 1,2,4 TRIAZOLES Public/Granted day:2010-12-23
Information query
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