Invention Grant
- Patent Title: Trisubstituted pyrazoles as acetylcholine receptor modulators
- Patent Title (中): 三取代吡唑作为乙酰胆碱受体调节剂
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Application No.: US12991119Application Date: 2009-05-08
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Publication No.: US08779158B2Publication Date: 2014-07-15
- Inventor: Johannes Wilhelmus John F. Thuring , Gregor James MacDonald , Wei Zhuang
- Applicant: Johannes Wilhelmus John F. Thuring , Gregor James MacDonald , Wei Zhuang
- Applicant Address: BE Beerse
- Assignee: Janssen Pharmaceutica NV
- Current Assignee: Janssen Pharmaceutica NV
- Current Assignee Address: BE Beerse
- Agent Peter Herridge
- Priority: EP08155991 20080509
- International Application: PCT/EP2009/055617 WO 20090508
- International Announcement: WO2009/135944 WO 20091112
- Main IPC: A61K31/4155
- IPC: A61K31/4155 ; A01N43/36 ; C07D231/02 ; C07D401/04

Abstract:
The present invention relates to 1-alkyl-3-aniline-5-aryl-pyrazole derivatives and pharmaceutically acceptable salts thereof, processes for preparing them, pharmaceutical compositions containing them and their use in therapy, according to Formula (I).The invention particularly relates to positive allosteric modulators of nicotinic acetylcholine receptors, such positive allosteric modulator having the capability to increase the efficacy of nicotinic receptor agonists.
Public/Granted literature
- US20110065683A1 TRISUBSTITUTED PYRAZOLES AS ACETYLCHOLINE RECEPTOR MODULATORS Public/Granted day:2011-03-17
Information query
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