Invention Grant
US08791265B2 Sulfonamido derivatives of 3,4-diarylpyrazoles as protein kinase inhibitors
有权
3,4-二芳基吡唑的磺酰胺衍生物作为蛋白激酶抑制剂
- Patent Title: Sulfonamido derivatives of 3,4-diarylpyrazoles as protein kinase inhibitors
- Patent Title (中): 3,4-二芳基吡唑的磺酰胺衍生物作为蛋白激酶抑制剂
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Application No.: US13574168Application Date: 2011-01-19
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Publication No.: US08791265B2Publication Date: 2014-07-29
- Inventor: Maurizio Pulici , Chiara Marchionni , Gabriella Traquandi
- Applicant: Maurizio Pulici , Chiara Marchionni , Gabriella Traquandi
- Applicant Address: IT Nerviano (MI)
- Assignee: Nerviano Medical Sciences S.R.L.
- Current Assignee: Nerviano Medical Sciences S.R.L.
- Current Assignee Address: IT Nerviano (MI)
- Agency: Brinks Gilson & Lione
- Priority: EP10151805 20100127
- International Application: PCT/EP2011/050654 WO 20110119
- International Announcement: WO2011/092088 WO 20110804
- Main IPC: C07D401/00
- IPC: C07D401/00 ; A61K31/44 ; A61K31/4439 ; C07D401/04

Abstract:
Compounds which are sulfonamido 3,4-diarylpyrazole derivatives, or pharmaceutically acceptable salts thereof, their preparation process and pharmaceutical compositions comprising them are disclosed; these compounds are useful in the treatment of diseases caused by and/or associated with an altered protein kinase activity such as cancer, viral infection, prevention of AIDS development in HIV-infected individuals, cell proliferative disorders, autoimmune and neurodegenerative disorders; also disclosed is their use as prodrugs.
Public/Granted literature
- US20130053419A1 SULFONAMIDO DERIVATIVES OF 3,4-DIARYLPYRAZOLES AS PROTEIN KINASE INHIBITORS Public/Granted day:2013-02-28
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