Invention Grant
US08822727B2 Processes for the preparation of intermediates related to the 5-HT2C agonist (R)-8-chloro-1-methyl-2,3,4,5-tetrahydro-1H-3-benzazepine
有权
制备与5-HT2C激动剂（R）-8-氯-1-甲基-2,3,4,5-四氢-1H-3-苯并氮杂相关的中间体的方法
- Patent Title: Processes for the preparation of intermediates related to the 5-HT2C agonist (R)-8-chloro-1-methyl-2,3,4,5-tetrahydro-1H-3-benzazepine
- Patent Title (中): 制备与5-HT2C激动剂（R）-8-氯-1-甲基-2,3,4,5-四氢-1H-3-苯并氮杂相关的中间体的方法
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Application No.: US12921101Application Date: 2009-03-03
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Publication No.: US08822727B2Publication Date: 2014-09-02
- Inventor: Marlon V. Carlos , Ryan O. Castro , Tawfik Gharbaoui , Xiao-Xiong Lu , You-An Ma , Nicholas D. San Martin
- Applicant: Marlon V. Carlos , Ryan O. Castro , Tawfik Gharbaoui , Xiao-Xiong Lu , You-An Ma , Nicholas D. San Martin
- Applicant Address: US CA San Diego
- Assignee: Arena Pharmaceuticals, Inc.
- Current Assignee: Arena Pharmaceuticals, Inc.
- Current Assignee Address: US CA San Diego
- International Application: PCT/US2009/001340 WO 20090303
- International Announcement: WO2009/111004 WO 20090911
- Main IPC: C07C211/00
- IPC: C07C211/00
Abstract:
The present invention provides processes and intermediates useful in the preparation of 8-chloro-1-methyl-2,3,4,5-tetrahydro-1H-3-benzazepine, a serotonin (5-HT) receptor agonist that is useful in the treatment or prophylaxis of, for example, central nervous system disorders, such as obesity.
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