Invention Grant
- Patent Title: Process for preparing docetaxel and its hydrate
- Patent Title (中): 多西紫杉醇及其水合物的制备方法
-
Application No.: US13634612Application Date: 2011-08-29
-
Publication No.: US08829210B2Publication Date: 2014-09-09
- Inventor: Vimal Kumar Shrawat , Rafiuddin , Veereshappa , Prashant Purohit
- Applicant: Vimal Kumar Shrawat , Rafiuddin , Veereshappa , Prashant Purohit
- Applicant Address: IN Raichure, Karnataka
- Assignee: Shilpa Medicare Limited
- Current Assignee: Shilpa Medicare Limited
- Current Assignee Address: IN Raichure, Karnataka
- Priority: IN1117/CHE/2011 20110401
- International Application: PCT/IN2011/000588 WO 20110829
- International Announcement: WO2012/131698 WO 20121004
- Main IPC: C07D305/14
- IPC: C07D305/14 ; A61K31/337

Abstract:
The present invention provide process of preparation of (2R,3S)—N-carboxy-3-phenylisoserine, N-tert-butyl ester, 13-ester with 5(β)-20-epoxy-1,2(α),4,7(β),10(β),13(α)-hexa hydroxy tax-11-en-9-one 4-acetate 2-benzoate or docetaxel and its trihydrate (I)
Public/Granted literature
- US20140039209A1 PROCESS FOR PREPARING DOCETAXEL AND ITS HYDRATE Public/Granted day:2014-02-06
Information query