Invention Grant
- Patent Title: Transdermally absorbable donepezil-containing preparation
- Patent Title (中): 透皮吸收多奈哌齐制剂
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Application No.: US13503198Application Date: 2010-10-18
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Publication No.: US08840922B2Publication Date: 2014-09-23
- Inventor: Satoshi Kawakami , Masahiro Yamaji
- Applicant: Satoshi Kawakami , Masahiro Yamaji
- Applicant Address: JP Higashikagawa-shi
- Assignee: Teikoku Seiyaku Co., Ltd.
- Current Assignee: Teikoku Seiyaku Co., Ltd.
- Current Assignee Address: JP Higashikagawa-shi
- Agency: Crowell & Moring LLP
- Priority: JP2009-242656 20091021
- International Application: PCT/JP2010/068260 WO 20101018
- International Announcement: WO2011/049038 WO 20110428
- Main IPC: A61K9/70
- IPC: A61K9/70 ; A61K31/445

Abstract:
Provided is a donepezil-containing transdermal absorption formulation that can sustainably administer donepezil for a long period of time, and can provide both a rapid increase in the blood level of donepezil and donepezil sustained release properties. The donepezil-containing transdermal absorption formulation is a transdermal absorption formulation produced by dissolving donepezil, which is the active ingredient, in an adhesive patch base that contains a hydrophobic polymer and an absorption promoter. The absorption promoter is one kind or two or more kinds selected from lauryl alcohol, triethyl citrate, isopropyl myristate, cetyl lactate, oleyl alcohol, sorbitan monooleate, polyethylene glycol monostearate, lauromacrogol, N-methyl-2-pyrrolidone, and triacetin.
Public/Granted literature
- US20120207816A1 Transdermally Absorbable Donepezil-Containing Preparation Public/Granted day:2012-08-16
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