Invention Grant
US08846665B2 6,7-dihydro-[1,3,4]thiadiazolo-[3,2-a][1,3]diazepin derivative and pharmaceutical composition containing the same as neuromuscular blocker or skeletal muscle relaxant, and method for the preparation
有权
6,7-二氢 - [1,3,4]噻二唑并[3,2-a] [1,3]二氮杂衍生物和含有神经肌肉阻滞剂或骨骼肌松弛剂的药物组合物及其制备方法
- Patent Title: 6,7-dihydro-[1,3,4]thiadiazolo-[3,2-a][1,3]diazepin derivative and pharmaceutical composition containing the same as neuromuscular blocker or skeletal muscle relaxant, and method for the preparation
- Patent Title (中): 6,7-二氢 - [1,3,4]噻二唑并[3,2-a] [1,3]二氮杂衍生物和含有神经肌肉阻滞剂或骨骼肌松弛剂的药物组合物及其制备方法
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Application No.: US14043401Application Date: 2012-04-11
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Publication No.: US08846665B2Publication Date: 2014-09-30
- Inventor: Adel S. El-Azab , Hussein I. El-Subbagh , Khalid A. Al-Rashood , Kamal E. H. El-Taher , Mohamed A. Al-Omar , Ghada S. Hassan , Fatmah A. Al-Omary , Alaa A. -M. Abdelaziz , Mohamed M. Hefnawy
- Applicant: Adel S. El-Azab , Hussein I. El-Subbagh , Khalid A. Al-Rashood , Kamal E. H. El-Taher , Mohamed A. Al-Omar , Ghada S. Hassan , Fatmah A. Al-Omary , Alaa A. -M. Abdelaziz , Mohamed M. Hefnawy
- Applicant Address: SA Riyadh
- Assignee: King Saud University
- Current Assignee: King Saud University
- Current Assignee Address: SA Riyadh
- Agency: Lucas & Mercanti, LLP
- Priority: EP11161597 20110408
- International Application: PCT/EP2012/001573 WO 20120411
- International Announcement: WO2012/136385 WO 20121011
- Main IPC: A61K31/55
- IPC: A61K31/55 ; C07D513/04
![6,7-dihydro-[1,3,4]thiadiazolo-[3,2-a][1,3]diazepin derivative and pharmaceutical composition containing the same as neuromuscular blocker or skeletal muscle relaxant, and method for the preparation](/abs-image/US/2014/09/30/US08846665B2/abs.jpg.150x150.jpg)
Abstract:
The present invention relates to a compound of formula 1 and addition salts thereof, a pharmaceutical composition containing the compound, a method for its preparation as well as the use of the compound as neuro-muscular blocker or skeletal muscle relaxant; wherein each symbol is as defined in the Specification.
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