Invention Grant
- Patent Title: Substituted pyrazine-2-carboxamide kinase inhibitors
- Patent Title (中): 取代的吡嗪-2-羧酰胺激酶抑制剂
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Application No.: US13684462Application Date: 2012-11-23
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Publication No.: US08877760B2Publication Date: 2014-11-04
- Inventor: Yonghong Song , Anjali Pandey
- Applicant: Portola Pharmaceuticals, Inc.
- Applicant Address: US CA South San Francisco
- Assignee: Portola Pharmaceuticals, Inc.
- Current Assignee: Portola Pharmaceuticals, Inc.
- Current Assignee Address: US CA South San Francisco
- Agency: Kilpatrick Townsend & Stockton LLP
- Main IPC: A61K31/427
- IPC: A61K31/427 ; A61K31/497 ; C07D241/20 ; C07D417/12

Abstract:
Provided are substituted pyrazine-2-carboxamide compounds of Formula I: useful for inhibiting of Syk kinase, intermediates used in making such compounds, methods for their preparation, pharmaceutical compositions thereof, methods for inhibition Syk kinase activity, and methods for treating conditions mediated at least in part by Syk kinase activity.
Public/Granted literature
- US20130131040A1 PYRAZINE KINASE INHIBITORS Public/Granted day:2013-05-23
Information query
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