Invention Grant
US08901302B2 Pyrazino[2,3-D]isoxazole derivative which is useful as a production intermediate of pyrazine carboxamide derivative
有权
吡嗪并[2,3-D]异恶唑衍生物，其可用作吡嗪甲酰胺衍生物的生产中间体
![Pyrazino[2,3-D]isoxazole derivative which is useful as a production intermediate of pyrazine carboxamide derivative](/docs/US/2014-12-02/US08901302B2/abs.jpg.600x600.jpg)
- Patent Title: Pyrazino[2,3-D]isoxazole derivative which is useful as a production intermediate of pyrazine carboxamide derivative
- Patent Title (中): 吡嗪并[2,3-D]异恶唑衍生物，其可用作吡嗪甲酰胺衍生物的生产中间体
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Application No.: US13886483Application Date: 2013-05-03
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Publication No.: US08901302B2Publication Date: 2014-12-02
- Inventor: Kouki Nakamura , Takeshi Murakami , Hiroyuki Naitou , Naoyuki Hanaki , Katsuyuki Watanabe
- Applicant: FUJIFILM Corporation , Toyama Chemical Co., Ltd.
- Applicant Address: JP Tokyo JP Tokyo
- Assignee: FUJIFILM Corporation,Toyama Chemical Co., Ltd.
- Current Assignee: FUJIFILM Corporation,Toyama Chemical Co., Ltd.
- Current Assignee Address: JP Tokyo JP Tokyo
- Agency: Sughrue Mion, PLLC
- Priority: JP2010-253414 20101112; JP2010-256510 20101117; JP2011-025760 20110209
- Main IPC: C07D241/50
- IPC: C07D241/50 ; C07C239/18 ; C07D498/04 ; C07C251/38 ; C07C255/23 ; C07C237/06 ; C07D261/18 ; C07C255/29 ; C07D241/18 ; C07D241/24
![Pyrazino[2,3-D]isoxazole derivative which is useful as a production intermediate of pyrazine carboxamide derivative](/abs-image/US/2014/12/02/US08901302B2/abs.jpg.150x150.jpg)
Abstract:
The object of the present invention is to provide a compound which is useful as a production intermediate of pyrazine carboxamide derivative such as 6-fluoro-3-hydroxy-2-pyrazine carboxamide. The present invention provides a pyrazino[2,3-d]isoxazole derivative represented by the formula (I): wherein X represents a halogen atom, a hydroxyl group or a sulfamoyloxy group, and Y represents —C(═O)R or —CN; wherein R represents a hydrogen atom, an alkoxy group an aryloxy group, an alkyl group, an aryl group or an amino group.
Public/Granted literature
- US20130245264A1 PYRAZINO[2,3-D]ISOXAZOLE DERIVATIVE Public/Granted day:2013-09-19
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