Invention Grant
US08933083B2 1,2,3-trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto such as diabetes and hyperglycemia
有权
1,2,3-三取代的芳基和杂芳基衍生物作为代谢的调节剂，以及与其相关的疾病的预防和治疗，如糖尿病和高血糖
- Patent Title: 1,2,3-trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto such as diabetes and hyperglycemia
- Patent Title (中): 1,2,3-三取代的芳基和杂芳基衍生物作为代谢的调节剂，以及与其相关的疾病的预防和治疗，如糖尿病和高血糖
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Application No.: US13618592Application Date: 2012-09-14
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Publication No.: US08933083B2Publication Date: 2015-01-13
- Inventor: Robert M. Jones , Graeme Semple , Beatriz Fioravanti , Guilherme Pereira , Imelda Calderon , Jane Laguerta Uy , Kameshwari Duvvuri , Jin Sun Karoline Choi , Yifeng Xiong , Vibha Dave , Mihai D. Azimioara
- Applicant: Robert M. Jones , Graeme Semple , Beatriz Fioravanti , Guilherme Pereira , Imelda Calderon , Jane Laguerta Uy , Kameshwari Duvvuri , Jin Sun Karoline Choi , Yifeng Xiong , Vibha Dave , Mihai D. Azimioara
- Applicant Address: US CA San Diego
- Assignee: Arena Pharmaceuticals, Inc.
- Current Assignee: Arena Pharmaceuticals, Inc.
- Current Assignee Address: US CA San Diego
- Agency: Fish & Richardson P.C.
- Agent Lyle W. Spruce
- Main IPC: C07D239/48
- IPC: C07D239/48 ; C07D401/14 ; C07D403/12 ; C07D403/14 ; C07D401/04 ; C07D401/12 ; C07D417/14 ; C07D409/14 ; C07D405/04 ; C07D419/14 ; C07D405/14 ; C07D213/79 ; C07D239/50 ; C07D213/68 ; C07D239/34 ; C07D411/14 ; C07D413/14 ; C07D295/096
Abstract:
The present invention relates to certain 1,2,3-trisubstituted aryl and heteroaryl derivatives of Formula (Ia) that are modulators of metabolism. Accordingly, compounds of the present invention are useful in the prophylaxis or treatment of metabolic disorders and complications thereof, such as, diabetes and obesity.
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