Invention Grant
- Patent Title: Macrocyclic compounds as Trk kinase inhibitors
- Patent Title (中): 大环化合物作为Trk激酶抑制剂
-
Application No.: US13698922Application Date: 2011-05-13
-
Publication No.: US08933084B2Publication Date: 2015-01-13
- Inventor: Steven Wade Andrews , Kevin Ronald Condroski , Julia Haas , Yutong Jiang , Gabrielle R. Kolakowski , Jeongbeob Seo , HongWoon Yang , Qian Zhao
- Applicant: Steven Wade Andrews , Kevin Ronald Condroski , Julia Haas , Yutong Jiang , Gabrielle R. Kolakowski , Jeongbeob Seo , HongWoon Yang , Qian Zhao
- Applicant Address: US CO Boulder
- Assignee: Array BioPharma Inc.
- Current Assignee: Array BioPharma Inc.
- Current Assignee Address: US CO Boulder
- Agency: Fish & Richardson P.C.
- International Application: PCT/US2011/036452 WO 20110513
- International Announcement: WO2011/146336 WO 20111124
- Main IPC: A61K31/519
- IPC: A61K31/519 ; C07D487/02 ; C07D519/00 ; C07D498/22 ; C07D487/04 ; C07D471/22

Abstract:
Compounds of Formula I: and pharmaceutically acceptable salts thereof, wherein ring A, ring B, W, m, D, R2, R2a, R3, R3a, and Z are as defined herein, are inhibitors of Trk kinases and are useful in the treatment of pain, cancer, inflammation, neurodegenerative diseases and certain infectious diseases.
Public/Granted literature
- US20130203776A1 MACROCYCLIC COMPOUNDS AS TRK KINASE INHIBITORS Public/Granted day:2013-08-08
Information query
IPC分类: