Invention Grant
US08975277B2 2,3-dihydrofuro[2,3-c]pyridin-2-ylpiperidine derivatives
有权
2,3-二氢呋喃并[2,3-c]吡啶-2-基哌啶衍生物
- Patent Title: 2,3-dihydrofuro[2,3-c]pyridin-2-ylpiperidine derivatives
- Patent Title (中): 2,3-二氢呋喃并[2,3-c]吡啶-2-基哌啶衍生物
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Application No.: US13911138Application Date: 2013-06-06
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Publication No.: US08975277B2Publication Date: 2015-03-10
- Inventor: Frank Himmelsbach , Elke Langkopf
- Applicant: Boehringer Ingelheim International GmbH
- Applicant Address: DE Ingelheim am Rhein
- Assignee: Boehringer Ingelheim International GmbH
- Current Assignee: Boehringer Ingelheim International GmbH
- Current Assignee Address: DE Ingelheim am Rhein
- Agent Michael P. Morris; Timothy X. Witkowski
- Priority: EP12171686 20120612
- Main IPC: A01N43/42
- IPC: A01N43/42 ; A61K31/44 ; A01N43/08 ; A61K31/34 ; C07D471/02 ; C07D307/87 ; C07D307/93 ; C07D491/048 ; C07D491/04
![2,3-dihydrofuro[2,3-c]pyridin-2-ylpiperidine derivatives](/abs-image/US/2015/03/10/US08975277B2/abs.jpg.150x150.jpg)
Abstract:
The present invention relates to compounds of general formula I, wherein the groups R1, LQ and Ar are as defined in the application, which have valuable pharmacological properties, and in particular bind to the GPR119 receptor and modulate its activity.
Public/Granted literature
- US20130331410A1 2,3-DIHYDROFURO[2,3-c]PYRIDIN-2-YLPIPERIDINE DERIVATIVES Public/Granted day:2013-12-12
Information query
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