Invention Grant
- Patent Title: Selective FAK inhibitors
- Patent Title (中): 选择性FAK抑制剂
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Application No.: US13542917Application Date: 2012-07-06
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Publication No.: US09120761B2Publication Date: 2015-09-01
- Inventor: Ian Peter Holmes , Ylva Bergman , Gillian Elizabeth Lunniss , Marica Nikac , Neil Chol , Catherine Fae Hemley , Scott Raymond Walker , Richard Charles Foitzik , Danny Ganame , Romina Lessene
- Applicant: Ian Peter Holmes , Ylva Bergman , Gillian Elizabeth Lunniss , Marica Nikac , Neil Chol , Catherine Fae Hemley , Scott Raymond Walker , Richard Charles Foitzik , Danny Ganame , Romina Lessene
- Applicant Address: AU Bundoora
- Assignee: Cancer Therapeutics CRC PTY LTD
- Current Assignee: Cancer Therapeutics CRC PTY LTD
- Current Assignee Address: AU Bundoora
- Agency: Holland & Knight LLP
- Agent W. David Wallace
- Main IPC: A61K31/506
- IPC: A61K31/506 ; C07D239/42 ; C07D403/12 ; C07D401/12 ; C07D401/14

Abstract:
A compound of the formula (I): where R1 or R2 is a cyclc amine group and R5 is an aromatic group with a carbonyl containing substituent for use as a FAK inhibitor.
Public/Granted literature
- US20130022594A1 SELECTIVE FAK INHIBITORS Public/Granted day:2013-01-24
Information query
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