Invention Grant
- Patent Title: Pharmaceutical composition for oral administration
- Patent Title (中): 用于口服给药的药物组合物
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Application No.: US12698566Application Date: 2010-02-02
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Publication No.: US09198904B2Publication Date: 2015-12-01
- Inventor: Takehiko Yasuji , Noriyuki Kinoshita , Hiroyuki Yoshino , Shuuya Kawahama , Kazuhiro Sako , Akio Sugihara
- Applicant: Takehiko Yasuji , Noriyuki Kinoshita , Hiroyuki Yoshino , Shuuya Kawahama , Kazuhiro Sako , Akio Sugihara
- Applicant Address: JP Tokyo
- Assignee: ASTELLAS PHARMA INC.
- Current Assignee: ASTELLAS PHARMA INC.
- Current Assignee Address: JP Tokyo
- Agency: Kilpatrick Townsend & Stockton LLP
- Main IPC: A61K31/47
- IPC: A61K31/47 ; A61K9/22 ; A61P13/02 ; A61K9/20 ; A61K9/48 ; A61K31/18 ; A61K31/439

Abstract:
The present invention relates to a pharmaceutical composition for oral administration comprising a modified release portion containing tamsulosin or a pharmaceutically acceptable salt thereof, and an immediate release portion containing solifenacin or a pharmaceutically acceptable salt thereof and a hydrophilic substance.In the pharmaceutical composition, the dissolution rate of each drug (in particular, solifenacin contained in the immediate release portion) is similar to those of the current single drug formulations, and the maximum percentage of drag dissolution of each drug (in particular, solifenacin contained in the immediate release portion) is 90% or more. Therefore, the pharmaceutical composition is a single formulation (i.e., a combined formulation) with a bioavailability equivalent to those of the current single drug formulations.
Public/Granted literature
- US20100233260A1 PHARMACEUTICAL COMPOSITION FOR ORAL ADMINISTRATION Public/Granted day:2010-09-16
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