Invention Grant
- Patent Title: Substituted pyrazolo[1,5-a]pyridines as JAK inhibitors
- Patent Title (中): 取代的吡唑并[1,5-a]吡啶作为JAK抑制剂
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Application No.: US13579344Application Date: 2011-02-18
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Publication No.: US09206183B2Publication Date: 2015-12-08
- Inventor: Jordi Bach Taña , Lluis Miquel Pages Santacana , Joan Taltavull Moll , Paul Robert Eastwood , Jacob Gonzalez Rodrigues , Victor Giulio Matassa
- Applicant: Jordi Bach Taña , Lluis Miquel Pages Santacana , Joan Taltavull Moll , Paul Robert Eastwood , Jacob Gonzalez Rodrigues , Victor Giulio Matassa
- Applicant Address: ES Barcelona
- Assignee: ALMIRALL, S.A.
- Current Assignee: ALMIRALL, S.A.
- Current Assignee Address: ES Barcelona
- Agency: Finnegan, Henderson, Farabow, Garrett & Dunner, L.L.P.
- Priority: EP10382039 20100218; EP10382217 20100805
- International Application: PCT/EP2011/000792 WO 20110218
- International Announcement: WO2011/101161 WO 20110825
- Main IPC: A61K31/437
- IPC: A61K31/437 ; C07D221/04 ; C07D487/04 ; A61K31/497 ; A61K31/4985 ; A61K31/506 ; A61K45/06 ; C07D471/04
![Substituted pyrazolo[1,5-a]pyridines as JAK inhibitors](/abs-image/US/2015/12/08/US09206183B2/abs.jpg.150x150.jpg)
Abstract:
New pyrazole derivatives having the chemical structure of formula (I) are disclosed; as well as process for their preparation, pharmaceutical compositions comprising them and their use in therapy as inhibitors of Janus Kinases (JAK).
Public/Granted literature
- US20140086870A9 PYRAZOLE DERIVATIVES AS JAK INHIBITORS Public/Granted day:2014-03-27
Information query
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