Invention Grant
- Patent Title: Thiazole derivatives
- Patent Title (中): 噻唑衍生物
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Application No.: US14118756Application Date: 2012-04-12
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Publication No.: US09249114B2Publication Date: 2016-02-02
- Inventor: Srinivasa R. Karra , Wolfgang Staehle , Eike Staub , Margarita Wucherer-Plietker
- Applicant: Srinivasa R. Karra , Wolfgang Staehle , Eike Staub , Margarita Wucherer-Plietker
- Applicant Address: DE Darmstadt
- Assignee: Merck Patent GmbH
- Current Assignee: Merck Patent GmbH
- Current Assignee Address: DE Darmstadt
- Agency: EMD Serono Research Institue
- Agent Thomas W. Brown
- International Application: PCT/US2012/033200 WO 20120412
- International Announcement: WO2012/161879 WO 20111129
- Main IPC: C07D417/04
- IPC: C07D417/04 ; C07D417/14 ; C07D413/14 ; C07D277/56 ; A61K31/426 ; A61K31/4439 ; A61K31/4545 ; A61K31/496 ; A61K31/5377 ; A61K45/06 ; A61N5/10
Abstract:
Compounds of the formula I in which R, R1, X and Y have the meanings indicated in Claim 1, are inhibitors of TBK1 and IKKε and can be employed, inter alia, for the treatment of cancer and inflammatory diseases.
Public/Granted literature
- US20140148457A1 Thiazole derivatives Public/Granted day:2014-05-29
Information query
