Invention Grant
- Patent Title: Compounds having antibacterial activity, process for their preparation and pharmaceutical compositions comprising them
- Patent Title (中): 具有抗菌活性的化合物,其制备方法和包含它们的药物组合物
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Application No.: US14371820Application Date: 2013-01-10
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Publication No.: US09255071B2Publication Date: 2016-02-09
- Inventor: Gerardo Burton , Fernando Javier Duran , Mario David Martinez , Elvira Zini , Veronica Mora Munoz , Lucila Bertoncello
- Applicant: Consejo Nacional de Investigaciones Cientificas y Técnicas (CONICET) , Laboratorios Richmond Sociedad Anónima Comercial Industrial y Financiera
- Applicant Address: AR Buenos Aires AR Buenos Aires
- Assignee: Consejo Nacional de Investigaciones Cientificas y Técnicas (CONICET),Laboratorios Richmond Sociedad Anónima Comercial Industrial y Financiera
- Current Assignee: Consejo Nacional de Investigaciones Cientificas y Técnicas (CONICET),Laboratorios Richmond Sociedad Anónima Comercial Industrial y Financiera
- Current Assignee Address: AR Buenos Aires AR Buenos Aires
- Agency: Greer, Burns & Crain, Ltd.
- Priority: AR20120100090 20120111
- International Application: PCT/IB2013/050235 WO 20130110
- International Announcement: WO2013/105053 WO 20130718
- Main IPC: C07D213/86
- IPC: C07D213/86 ; C07C235/34 ; C07C51/60 ; C07C231/02 ; C07C235/38 ; C07C51/347 ; C07C259/08 ; C07D213/81 ; C07D295/185

Abstract:
A pharmaceutically acceptable salt, prodrug or derivative compound of the formula I, wherein R1 is selected from H, a (C1-C5) alkyl group and a COR4 group; R2 is selected from H, a (C1-C5) alkyl group and a COR5 group; R3 is selected from H, a (C1-C5) alkyl group, a (C1-C5)-O-alkyl group, a cycloalkyl of (C5-C6) carbon atoms, an aryl group, and an aryl (C1-C5) alkyl group wherein the aryl group can be an unsubstituted aryl or substituted with one or more R6 groups and an NHCOR5 group, or the R2 and R3 groups together with N may form a piperidine, morpholine or piperazine group; R4 is selected from H and a (C1-C5)alkyl group; R5 is selected from an aryl group unsubstituted or substituted with one or more R6, linear or branched(C1-C5) alkyl or pyridyne groups and a pyridine group; R6 is selected from (C1-C5)alkyl groups, halogen and nitro.
Public/Granted literature
Information query
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