Invention Grant
- Patent Title: Heterocyclic compounds as bromodomain inhibitors
- Patent Title (中): 杂环化合物作为溴结构域抑制剂
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Application No.: US14134793Application Date: 2013-12-19
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Publication No.: US09271978B2Publication Date: 2016-03-01
- Inventor: Shuang Liu , Bryan Cordell Duffy , John Frederick Quinn , May Xiaowu Jiang , Ruifang Wang , Gregory Scott Martin , He Zhao , Bruce Francis Molino , Peter Ronald Young
- Applicant: Shuang Liu , Bryan Cordell Duffy , John Frederick Quinn , May Xiaowu Jiang , Ruifang Wang , Gregory Scott Martin , He Zhao , Bruce Francis Molino , Peter Ronald Young
- Applicant Address: CA Calgary, Alberta
- Assignee: Zenith Epigenetics Corp.
- Current Assignee: Zenith Epigenetics Corp.
- Current Assignee Address: CA Calgary, Alberta
- Agency: Finnegan, Henderson, Farabow, Garrett & Dunner, LLP
- Main IPC: A61K31/501
- IPC: A61K31/501 ; C07D413/04 ; C07D401/12 ; A61K31/4439 ; C07D417/04 ; C07D413/14 ; A61K31/496 ; C07D237/04 ; A61K31/50 ; A61K45/06

Abstract:
The present disclosure relates to compounds, which are useful for inhibition of BET protein function by binding to bromodomains, and their use in therapy.
Public/Granted literature
- US20140179648A1 Novel Heterocyclic Compounds as Bromodomain Inhibitors Public/Granted day:2014-06-26
Information query
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