Invention Grant
US09303052B2 Water-soluble benzoazepine compound and its pharmaceutical composition
有权
水溶性苯并吖庚因化合物及其药物组成
- Patent Title: Water-soluble benzoazepine compound and its pharmaceutical composition
- Patent Title (中): 水溶性苯并吖庚因化合物及其药物组成
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Application No.: US13964853Application Date: 2013-08-12
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Publication No.: US09303052B2Publication Date: 2016-04-05
- Inventor: Makoto Komatsu , Fumitaka Goto , Yasuhiro Menjo , Keigo Yamada , Takakuni Matsuda , Yusuke Kato
- Applicant: Otsuka Pharmaceutical Co., Ltd.
- Applicant Address: JP Tokyo
- Assignee: I. OTSUKA PHARMACEUTICAL CO., LTD.
- Current Assignee: I. OTSUKA PHARMACEUTICAL CO., LTD.
- Current Assignee Address: JP Tokyo
- Agency: Finnegan, Henderson, Farabow, Garrett & Dunner, L.L.P.
- Priority: JP2005-375457 20051227
- Main IPC: C07F9/553
- IPC: C07F9/553
Abstract:
The present invention provides a benzoazepine compound represented by following general formula (1): or a salt thereof, wherein R represents a hydrogen atom, a hydroxy group optionally protected with a protecting group, etc., R1 represents a hydrogen atom or hydroxy-protecting group, and X represents an oxygen atom or a sulfur atom. The benzoazepine compound of the present invention and salts thereof have high solubility in water, and can be suitably used for injections.
Public/Granted literature
- US20130331358A1 Water-Soluble Benzoazepine Compound and Its Pharmaceutical Composition Public/Granted day:2013-12-12
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