Invention Grant
US09315463B2 Cyclohexylamine derivatives having β2 adrenergic agonist and M3 muscarinic antagonist activities
有权
具有二肾上腺素能激动剂和M3毒蕈碱拮抗剂活性的环己胺衍生物
- Patent Title: Cyclohexylamine derivatives having β2 adrenergic agonist and M3 muscarinic antagonist activities
- Patent Title (中): 具有二肾上腺素能激动剂和M3毒蕈碱拮抗剂活性的环己胺衍生物
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Application No.: US13697060Application Date: 2011-05-13
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Publication No.: US09315463B2Publication Date: 2016-04-19
- Inventor: Maria Prat Quinones , Silvia Fonquerna Pou , Carlos Puig Duran , Wenceslao Lumeras Amador , Jose Aiguade Bosch , Juan Francisco Caturla Jovaloyes
- Applicant: Maria Prat Quinones , Silvia Fonquerna Pou , Carlos Puig Duran , Wenceslao Lumeras Amador , Jose Aiguade Bosch , Juan Francisco Caturla Jovaloyes
- Applicant Address: ES Barcelona
- Assignee: Almirall, S.A.
- Current Assignee: Almirall, S.A.
- Current Assignee Address: ES Barcelona
- Agency: Finnegan, Henderson, Farabow, Garrett & Dunner
- Priority: EP10382118 20100513
- International Application: PCT/EP2011/002376 WO 20110513
- International Announcement: WO2011/141180 WO 20111117
- Main IPC: C07D215/26
- IPC: C07D215/26 ; C07D409/14 ; A61K31/4709 ; B29C44/12

Abstract:
The present disclosure relates to novel compounds having β2 adrenergic agonist and M3 muscarinic antagonist dual activity, to pharmaceutical compositions containing them, to the process for their preparation and to their use in respiratory therapies.
Public/Granted literature
- US20130281415A9 NEW CYCLOHEXYLAMINE DERIVATIVES HAVING ß2 ADRENERGIC AGONIST AND M3 MUSCARINIC ANTAGONIST ACTIVITIES Public/Granted day:2013-10-24
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