Invention Grant
- Patent Title: Aldehyde derivative of substitute oxazolidinones
- Patent Title (中): 取代恶唑烷酮的醛衍生物
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Application No.: US14436018Application Date: 2013-12-24
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Publication No.: US09359341B2Publication Date: 2016-06-07
- Inventor: Nitin Sharadchandra Pradhan , Nilesh Sudhir Patil , Rajesh Ramchandra Walavalkar , Nilesh Subhas Kulkarni , Sandip Babanrao Pawar , Tarak Sambhaji Pawar
- Applicant: WANBURY LTD.
- Applicant Address: unknown Navi Mumbai, Maharashtra
- Assignee: WANBURY LTD.
- Current Assignee: WANBURY LTD.
- Current Assignee Address: unknown Navi Mumbai, Maharashtra
- Agency: Locke Lord LLP
- Agent Tim Tingkang Xia, Esq.
- Priority: IN3359/MUM/2012 20121226
- International Application: PCT/IN2013/000801 WO 20131224
- International Announcement: WO2014/102822 WO 20140703
- Main IPC: A61K31/5377
- IPC: A61K31/5377 ; C07D413/14 ; C07D413/10

Abstract:
The present invention relates to the prodrug of 5-chloro-N-({(5S)-2-oxo-3-[4-(3-oxo-morpholin-4-yl)phenyl]-1,3-oxazolidin-5-yl}methyl)thiophene-2-carboxamide, rivaroxaban per se; processes for their preparation, and the application in treatment and/or prophylaxis of diseases, especially of thromboembolic disorders. The prodrug of a compound of formula (B) is chemically designated as 5-chloro-N-formyl-N-({(5S)-2-oxo-3-[4-(3-oxomorpholin-4-yl)phenyl]-1,3-oxazolidin-5-yl}methyl)thiophene-2-carboxamide.
Public/Granted literature
- US20150259333A1 ALDEHYDE DERIVATIVE OF SUBSTITUTE OXAZOLIDINONES Public/Granted day:2015-09-17
Information query
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