Invention Grant
US09388188B2 Synthetic route for the preparation of β-aminobutyryl substituted 5,6,7,8-tetrahydro[1,4]diazolo[4,3-alpha ]pyrazin-7-yl compounds
有权
用于制备&b-氨基丁酰基取代的5,6,7,8-四氢[1,4]二唑并[4,3-a]吡嗪-7-基化合物的合成路线
- Patent Title: Synthetic route for the preparation of β-aminobutyryl substituted 5,6,7,8-tetrahydro[1,4]diazolo[4,3-alpha ]pyrazin-7-yl compounds
- Patent Title (中): 用于制备&b-氨基丁酰基取代的5,6,7,8-四氢[1,4]二唑并[4,3-a]吡嗪-7-基化合物的合成路线
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Application No.: US14406686Application Date: 2013-06-13
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Publication No.: US09388188B2Publication Date: 2016-07-12
- Inventor: Stefan Starcevic , Peter Mrak , Gregor Kopitar
- Applicant: Lek Pharmaceuticals d.d.
- Applicant Address: SI
- Assignee: Lek Pharmaceuticals d.d.
- Current Assignee: Lek Pharmaceuticals d.d.
- Current Assignee Address: SI
- Agency: Luedeka Neely Group, P.C.
- Priority: EP12172012 20120614
- International Application: PCT/EP2013/062307 WO 20130613
- International Announcement: WO2013/186326 WO 20131219
- Main IPC: C07D487/04
- IPC: C07D487/04 ; C07D205/08 ; C07C227/18
![Synthetic route for the preparation of β-aminobutyryl substituted 5,6,7,8-tetrahydro[1,4]diazolo[4,3-alpha ]pyrazin-7-yl compounds](/abs-image/US/2016/07/12/US09388188B2/abs.jpg.150x150.jpg)
Abstract:
The present invention relates to a process for preparing □-aminobutyryl substituted 5,6,7,8-tetrahydro[1,4]diazolo[4,3-α]pyrazin-7-yl compounds.
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