Invention Grant
- Patent Title: Process for preparing benzofuran-2-carboxamide derivatives
- Patent Title (中): 制备苯并呋喃-2-甲酰胺衍生物的方法
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Application No.: US14410198Application Date: 2013-07-01
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Publication No.: US09399630B2Publication Date: 2016-07-26
- Inventor: Mohan Rao Dodda , Jithender Aadepu
- Applicant: SYMED LABS LIMITED
- Applicant Address: IN
- Assignee: Symed Labs Limited
- Current Assignee: Symed Labs Limited
- Current Assignee Address: IN
- Agency: Caesar Rivise, PC
- Priority: IN2629/CHE/2012 20120702
- International Application: PCT/IN2013/000404 WO 20130701
- International Announcement: WO2014/006637 WO 20140109
- Main IPC: C07D319/06
- IPC: C07D319/06 ; C07D307/85 ; C07D401/12 ; C07D209/12 ; C07D209/10

Abstract:
Provided herein are novel, commercially viable and industrially advantageous processes for the preparation of benzofuran-2-carboxamide derivatives and their intermediates, or a pharmaceutically acceptable salt thereof, in high yield and purity. Provided particularly herein are novel, commercially viable and industrially advantageous processes for the preparation of vilazodone or a pharmaceutically acceptable salt thereof in high yield and purity. Provided also herein is an improved and commercially viable process for the preparation of 3-(4-hydroxybutyl)-1H-indole-5-carbonitrile, in high yield and purity, using novel intermediate compound 3-(4-hydroxybutyryl)-1H-indole-5-carbonitrile.
Public/Granted literature
- US20150322030A1 IMPROVED PROCESS FOR PREPARING BENZOFURAN-2-CARBOXAMIDE DERIVATIVES Public/Granted day:2015-11-12
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