Invention Grant
US09403835B2 Tetraaza-cyclopenta[a]indenyl and their use as positive allosteric modulators
有权
四环 - 环戊二烯并[a]茚基,它们用作正变构调节剂
- Patent Title: Tetraaza-cyclopenta[a]indenyl and their use as positive allosteric modulators
- Patent Title (中): 四环 - 环戊二烯并[a]茚基,它们用作正变构调节剂
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Application No.: US14366901Application Date: 2012-11-30
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Publication No.: US09403835B2Publication Date: 2016-08-02
- Inventor: Dominique Swinnen , Cyril Montagne , Vincent Pomel , Anna Quattropani , Jerome Molette , Patrick Gerber
- Applicant: Merck Patent GmbH
- Applicant Address: CH Aubonne
- Assignee: Ares Trading S.A.
- Current Assignee: Ares Trading S.A.
- Current Assignee Address: CH Aubonne
- Agency: EMD Serono Research and Development Institute
- Agent Dwight D. Kim
- Priority: EP11195214 20111222; EP12171415 20120611
- International Application: PCT/EP2012/004968 WO 20121130
- International Announcement: WO2013/091773 WO 20130627
- Main IPC: A61K31/519
- IPC: A61K31/519 ; C07D487/14 ; C07D471/14 ; C07D519/00 ; A61K31/5513
![Tetraaza-cyclopenta[a]indenyl and their use as positive allosteric modulators](/abs-image/US/2016/08/02/US09403835B2/abs.jpg.150x150.jpg)
Abstract:
The present invention provides compounds of Formula (I) as M1 receptor positive allosteric modulators for the treatment of diseases mediated by the muscarinic M1 mediator.
Public/Granted literature
- US20150018343A1 Tetraaza-cyclopenta[a]indenyl and their use as Positive Allosteric Modulators Public/Granted day:2015-01-15
Information query
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