Invention Grant
- Patent Title: Crystalline salts of asenapine
- Patent Title (中): 阿替那磷的结晶盐
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Application No.: US14113091Application Date: 2012-04-30
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Publication No.: US09447109B2Publication Date: 2016-09-20
- Inventor: Samuele Frigoli , Davide Longoni , Tamara Danelli , Marco Alpegiani
- Applicant: Samuele Frigoli , Davide Longoni , Tamara Danelli , Marco Alpegiani
- Applicant Address: IT Rodano
- Assignee: OLON S.P.A.
- Current Assignee: OLON S.P.A.
- Current Assignee Address: IT Rodano
- Agency: Silvia Salvadori, PC.
- Agent Silvia Salvadori
- Priority: ITMI2011A0734 20110502
- International Application: PCT/IB2012/052151 WO 20120430
- International Announcement: WO2012/150538 WO 20121108
- Main IPC: C07D491/044
- IPC: C07D491/044

Abstract:
Disclosed is asenapine phosphate of formula (I) and its enantiomer (I) which can be used to prepare asenapine maleate. Further disclosed is a monoclinic crystalline form of asenapine maleate.
Public/Granted literature
- US20140051741A1 CRYSTALLINE SALTS OF ASENAPINE Public/Granted day:2014-02-20
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