Invention Grant
US09533953B2 Method of preparation of crystal forms of 4-(cyclopropylmethoxy)-n-(3,5-dichloro-1-oxidopyridyn-4-yl)-5-methoxypyridine-2-carboxamide and crystal forms thereof 有权
制备4-(环丙基甲氧基) - 正 - (3,5-二氯-1-氧基吡啶-4-基)-5-甲氧基吡啶-2-甲酰胺及其晶体形式的晶型的方法

  • Patent Title: Method of preparation of crystal forms of 4-(cyclopropylmethoxy)-n-(3,5-dichloro-1-oxidopyridyn-4-yl)-5-methoxypyridine-2-carboxamide and crystal forms thereof
  • Patent Title (中): 制备4-(环丙基甲氧基) - 正 - (3,5-二氯-1-氧基吡啶-4-基)-5-甲氧基吡啶-2-甲酰胺及其晶体形式的晶型的方法
  • Application No.: US14647799
    Application Date: 2013-11-28
  • Publication No.: US09533953B2
    Publication Date: 2017-01-03
  • Inventor: Pascal BillotDidier BrigeAlexandre GiulianiHagit ElmalehMarc-Antoine Perrin
  • Applicant: SANOFI
  • Applicant Address: FR Paris
  • Assignee: SANOFI
  • Current Assignee: SANOFI
  • Current Assignee Address: FR Paris
  • Agency: Morrison & Foerster LLP
  • Priority: EP12306479 20121128
  • International Application: PCT/EP2013/074972 WO 20131128
  • International Announcement: WO2014/083107 WO 20140605
  • Main IPC: C07D213/89
  • IPC: C07D213/89
Method of preparation of crystal forms of 4-(cyclopropylmethoxy)-n-(3,5-dichloro-1-oxidopyridyn-4-yl)-5-methoxypyridine-2-carboxamide and crystal forms thereof
Abstract:
The present invention relates to a process of preparation of Crystal Forms of 4-(cyclopropylmethoxy)-N-(3,5-dichloro-1-oxidopyridin-4-yl)-5-methoxypyridine-2-carboxamide of formula (I), said Crystal Forms which are designated as Crystal Forms A to I A and their use as a medicament.
Information query
Patent Agency Ranking
0/0