Invention Grant
- Patent Title: Bicyclic heterocycles as FGFR inhibitors
- Patent Title (中): 双环杂环作为FGFR抑制剂
-
Application No.: US14256438Application Date: 2014-04-18
-
Publication No.: US09533984B2Publication Date: 2017-01-03
- Inventor: Yaping Sun , Liang Lu , Wenqing Yao , Jincong Zhuo , Liangxing Wu , Meizhong Xu , Ding-Quan Qian , Chunhong He , Fenglei Zhang
- Applicant: Incyte Corporation , Incyte Holdings Corporation
- Applicant Address: US DE Wilmington US DE Wilmington
- Assignee: Incyte Holdings Corporation,Incyte Corporation
- Current Assignee: Incyte Holdings Corporation,Incyte Corporation
- Current Assignee Address: US DE Wilmington US DE Wilmington
- Agency: Fish & Richardson P.C.
- Main IPC: C07D471/04
- IPC: C07D471/04 ; A61P35/00 ; A61K31/4375

Abstract:
The present invention relates to bicyclic heterocycles, and pharmaceutical compositions of the same, that are inhibitors of one or more FGFR enzymes and are useful in the treatment of FGFR-associated diseases such as cancer.
Public/Granted literature
- US20140315902A1 BICYCLIC HETEROCYCLES AS FGFR INHIBITORS Public/Granted day:2014-10-23
Information query