Invention Grant
- Patent Title: Pyridine carboxylic acid based compound used as a P2X1 and P2X3 receptor antagonist, a production method for the same and a composition comprising the same
- Patent Title (中): 用作P2X1和P2X3受体拮抗剂的吡啶羧酸类化合物及其制备方法及其组合物
-
Application No.: US13643674Application Date: 2010-12-20
-
Publication No.: US09546139B2Publication Date: 2017-01-17
- Inventor: Yong-Chul Kim , Kwan-Young Jung , Joong Heui Cho
- Applicant: Yong-Chul Kim , Kwan-Young Jung , Joong Heui Cho
- Applicant Address: KR Buk-gu, Gwangju
- Assignee: GWANGJU INSTITUTE OF SCIENCE AND TECHNOLOGY
- Current Assignee: GWANGJU INSTITUTE OF SCIENCE AND TECHNOLOGY
- Current Assignee Address: KR Buk-gu, Gwangju
- Agency: Nath, Goldberg & Meyer
- Agent Joshua B. Goldberg; Tanya E. Harkins
- Priority: KR10-2010-0038535 20100426
- International Application: PCT/KR2010/009096 WO 20101220
- International Announcement: WO2011/136459 WO 20111103
- Main IPC: C07D213/79
- IPC: C07D213/79 ; C07D213/77 ; C07D213/80 ; C07D213/65 ; C07D213/66
Abstract:
Provided are a novel pyridine carboxylic acid based compound used as a P2X1 and P2X3 receptor antagonist, a production method for the same and a composition comprising the same. The compound according to the present invention is a powerful antagonist of P2X1 and P2X3 receptors, and hence can be used as a drug for treating or preventing diseases involving neurological pain or chronic inflammatory diseases which are diseases caused by P2X1 and P2X3 receptor activity.
Public/Granted literature
Information query
IPC分类:
